SCHEMBL6708336

SCHEMBL6708336

NC(=O)c1c[nH]c2ccsc2c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.49
HTR3A P46098 1/20 0.49
ALDH1A1 P00352 4/20 0.45
ATM Q13315 1/20 0.45
MAPT P10636 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPK1 P28482 1/20 0.42
MAPK8 P45983 1/20 0.39
PARP1 P09874 1/20 0.38
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
PTK2 Q05397 1/20 0.36
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
MAPK10 P53779 2/20 0.33
HTT P42858 1/20 0.33
PDPK1 O15530 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15562633 0.88 ALDH1A1 (0.49) CYP3A4HTR3AALDH1A1ATMMAPT
SCHEMBL2793777 0.85 CYP3A4 (0.50) CYP3A4HTR3AALDH1A1MAPTMEN1
SCHEMBL13229697 0.83 CYP3A4 (0.49) CYP3A4HTR3AALDH1A1MAPTMEN1
SCHEMBL13229581 0.80 CYP3A4 (0.55) CYP3A4HTR3AALDH1A1MAPTKMT2A
SCHEMBL10472393 0.77 GABRA1 (0.52) CYP3A4HTR3AHTR2AHTR2CHTR2B
SCHEMBL31549260 0.75 F7 (0.43) CYP3A4HTR3AALDH1A1MAPTMEN1
SCHEMBL13229587 0.75 CFTR (0.63) CYP3A4HTR3AALDH1A1MEN1KMT2A
SCHEMBL6332699 0.73 ALDH1A1 (0.42) ALDH1A1ATMMAPTMEN1KMT2A
SCHEMBL6479523 0.72 POLB (0.56) CYP3A4HTR3AKMT2ANPC1RAB9A
SCHEMBL13229624 0.71 CFTR (0.48) CYP3A4HTR3AALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040248927-A1 Preventive agent/remedial agent for constipation predominant ibs MITSUBISHI PHARMA CORPORATION (JP) 2004-12-09 US disclosed
EP-0269295-A1 Therapeutic agents The Boots Company PLC (GB) 1988-06-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248927-A1 Preventive agent/remedial agent for constipation predominant ibs BRS3, SLC10A2, FABP2 CYP3A4 2819/4885HTR3A 25/4885ALDH1A1 1982/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.