SCHEMBL6715150

SCHEMBL6715150

CCOC(=O)C(Cc1ccc(OCCNC(=O)c2ccc(-c3ccc(F)cc3)cc2)cc1)Oc1ccc(C(C)C)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 4/20 0.48
PPARG P37231 3/20 0.46
EPHX2 P34913 1/20 0.46
ALDH1A1 P00352 2/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 4/20 0.45
MAPT P10636 3/20 0.45
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PPARA Q07869 1/20 0.40
GCG P01275 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6716576 0.92 PPARG (0.46) HCAR2PPARGRAB9ANPC1MAPT
SCHEMBL6716263 0.92 NPC1 (0.53) HCAR2PPARGEPHX2ALDH1A1RAB9A
SCHEMBL6714779 0.91 RAB9A (0.48) PPARGEPHX2ALDH1A1RAB9ANPC1
SCHEMBL6716087 0.91 HCAR2 (0.48) HCAR2PPARGEPHX2ALDH1A1RAB9A
SCHEMBL6715892 0.90 PPARG (0.52) HCAR2PPARGALDH1A1RAB9ANPC1
SCHEMBL6713067 0.87 NPC1 (0.45) HCAR2EPHX2ALDH1A1RAB9ANPC1
SCHEMBL6715977 0.87 PPARA (0.50) HCAR2PPARGEPHX2ALDH1A1RAB9A
SCHEMBL6713405 0.86 GCG (0.44) HCAR2PPARGRAB9ANPC1MAPT
SCHEMBL6713127 0.85 NPC1 (0.52) PPARGRAB9ANPC1MAPTSMN1; SMN2
SCHEMBL6715209 0.85 GCG (0.51) HCAR2EPHX2ALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040006141-A1 Amidocarboxylic acid compounds SANKYO COMPANY, LTD (JP) 2004-01-08 US disclosed
US-6528525-B1 Amidocarboxylic acid derivatives SANKYO COMPANY, LIMITED (JP) 2003-03-04 US disclosed
EP-1026149-A1 AMIDOCARBOXYLIC ACID DERIVATIVES Sankyo Company Limited (JP) 2000-08-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040006141-A1 Amidocarboxylic acid compounds NR1H2, AGK, APOL1 HCAR2 429/4885PPARG 23/4885EPHX2 3288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.