SCHEMBL6715302

SCHEMBL6715302

CC(C)(C)OC(=O)N(Cc1ccccc1)[C@H]1C2CN(c3ccc(NC(=O)OCc4ccccc4)cc3F)C[C@@H]21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.44
BACE1 P56817 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
MAPT P10636 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
ATM Q13315 1/20 0.39
MGLL Q99685 2/20 0.39
UBE2M P61081 2/20 0.38
DCUN1D1 Q96GG9 2/20 0.38
NPY2R P49146 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP2C9 P11712 1/20 0.38
PKM P14618 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5464908 1.00 RORC (0.44) RORCBACE1PTGDR2MAPTNPC1
SCHEMBL5463410 0.90 RORC (0.42) RORCBACE1PTGDR2MAPTNPC1
SCHEMBL5746506 0.87 RORC (0.42) RORCBACE1NPC1RAB9AMGLL
SCHEMBL6477484 0.85 RORC (0.51) RORCPTGDR2MAPTNPC1RAB9A
SCHEMBL6477875 0.85 RORC (0.46) RORCPTGDR2MAPTNPC1RAB9A
SCHEMBL6711562 0.83 RORC (0.39) RORCBACE1NPC1RAB9AMGLL
SCHEMBL5744670 0.83 RORC (0.39) RORCBACE1NPC1RAB9AMGLL
SCHEMBL5466676 0.83 HSD11B1 (0.41) RORCMAPTSMN1; SMN2ALDH1A1TP53
SCHEMBL5461178 0.80 ALDH1A1 (0.44) MAPTALDH1A1MEN1KMT2A
SCHEMBL6510132 0.78 NPY2R (0.52) BACE1PTGDR2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385834-A1 BICYCLO[3,1,0]HEXANE CONTAINING OXAZOLIDINONE ANTIBIOTIC AND DERIVATIVES THEREOF Merck & Co., Inc. (US) 2004-02-04 EP disclosed
WO-2003027083-A1 BICYCLO[3,1,0]HEXANE CONTAINING OXAZOLIDINONE ANTIBIOTIC AND DERIVATIVES THEREOF MERCK & CO., INC. (US) 2003-04-03 WO disclosed