SCHEMBL6716320

SCHEMBL6716320

NC(=O)N1CCN(c2ccccc2Cl)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.62
HTR7 P34969 2/20 0.57
HTR1A P08908 2/20 0.57
HTR2A P28223 1/20 0.57
HTR6 P50406 1/20 0.57
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
GAA P10253 2/20 0.56
ALDH1A1 P00352 2/20 0.56
NPSR1 Q6W5P4 2/20 0.56
GLA P06280 1/20 0.56
MAPT P10636 1/20 0.55
MAPK1 P28482 3/20 0.54
RAB9A P51151 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
GRM5 P41594 1/20 0.54
KDM4E B2RXH2 1/20 0.51
ADRB1 P08588 1/20 0.50
LMNA P02545 1/20 0.50
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30965800 0.88 DRD2 (0.58) AKR1C3HTR7HTR1AHTR2AHTR6
SCHEMBL2857040 0.84 AKR1C3 (0.64) AKR1C3HTR7HTR1AMEN1KMT2A
SCHEMBL17276412 0.84 AKR1C3 (0.64) AKR1C3HTR7HTR1AMEN1KMT2A
SCHEMBL9565829 0.82 AKR1C3 (0.62) AKR1C3HTR7MEN1KMT2AGAA
SCHEMBL3436755 0.81 AKR1C3 (0.63) AKR1C3MEN1KMT2AALDH1A1ADRB1
SCHEMBL28396664 0.80 ADRB1 (0.71) AKR1C3HTR1AALDH1A1RAB9AKDM4E
Hydrochloric Acid SCHEMBL6987606 0.80 GRM5 (0.59) AKR1C3HTR7MEN1KMT2AGAA
SCHEMBL8274961 0.80 ADAM10 (0.55) AKR1C3HTR7MEN1KMT2AGAA
SCHEMBL23064287 0.79 GAA (0.67) AKR1C3HTR2AMEN1KMT2AGAA
SCHEMBL21987068 0.79 MEN1 (0.72) AKR1C3HTR1AHTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1146790-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-03-17 EP claimed
JP-2002535256-A 2002-10-22 JP claimed
EP-1146790-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2001-10-24 EP claimed
WO-2000042852-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-27 WO claimed
EP-1313477-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-03-03 EP disclosed
EP-1313477-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2003-05-28 EP disclosed
WO-2002005819-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2002-01-24 WO disclosed