SCHEMBL671737

SCHEMBL671737

CC(C)(C)c1n[nH]c(CN(C(=O)O)C(C)(C)C)n1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL672749 0.88 TDP1 (0.31) TDP1MEN1KMT2AHTTL3MBTL1
SCHEMBL5116803 0.74 ROCK2 (0.50)
SCHEMBL25244288 0.71 MEN1 (0.33) TDP1MEN1KMT2AHTTL3MBTL1
SCHEMBL9912664 0.68 RAB9A (0.36) HTTSMN1; SMN2
SCHEMBL7478096 0.67 MEN1 (0.50) TDP1MEN1KMT2AMAPT
SCHEMBL16616069 0.66 MEN1 (0.40) TDP1MEN1KMT2AHTTL3MBTL1
SCHEMBL18905841 0.65 GLA (0.41) MEN1KMT2AMAPT
SCHEMBL20115738 0.65 CGAS (0.42) KMT2AMAPT
SCHEMBL17094558 0.65 KDM6B (0.44) HTTL3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL17094136 0.65 ALDH1A1 (0.34) TDP1MEN1KMT2AHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606033-A1 SUBSTITUTED CYCLIC CARBOXAMIDE AND UREA DERIVATIVES AS LIGANDS OF THE VANILLOID RECEPTOR Grünenthal GmbH (DE) 2013-06-26 EP disclosed
WO-2012022487-A1 SUBSTITUTED CYCLIC CARBOXAMIDE AND UREA DERIVATIVES AS LIGANDS OF THE VANILLOID RECEPTOR Grünenthal GmbH (DE) 2012-02-23 WO disclosed