SCHEMBL6722707

SCHEMBL6722707

CS(=O)(=O)c1ccc(-c2c(-c3ccc(Cl)c(Cl)c3)noc2C(F)F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.41
LMNA P02545 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PTGS1 P23219 1/20 0.35
CSNK1D P48730 2/20 0.33
MAPK14 Q16539 2/20 0.33
SCN9A Q15858 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6722948 0.93 PTGS2 (0.43) PTGS2PTGS1TRPV1PIK3CDPIK3CA
SCHEMBL7042225 0.92 PTGS2 (0.43) PTGS2PTGS1CSNK1DMAPK14PIK3CD
SCHEMBL6723359 0.89 CA1 (0.39) PTGS2PTGS1
SCHEMBL6722959 0.89 PTGS2 (0.43) PTGS2NPSR1CSNK1DMAPK14MAPK9
SCHEMBL6721360 0.89 PTGS2 (0.40) PTGS2CSNK1DMAPK14MAPK9MAPK10
SCHEMBL6722585 0.89 PAX8 (0.40) PTGS2SCN9A
SCHEMBL6723642 0.89 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL6725529 0.89 PTGS2 (0.38) PTGS2PTGS1CSNK1DMAPK14MAPK9
SCHEMBL6729625 0.88 PTGS2 (0.42) PTGS2LMNANPSR1PTGS1CSNK1D
SCHEMBL6719025 0.87 PTGS2 (0.43) PTGS2PTGS1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040092552-A1 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation PHARMACIA CORPORATION 2004-05-13 US disclosed
EP-1296971-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2003-04-02 EP disclosed
US-20020183362-A1 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation PHARMACIA CORPORATION 2002-12-05 US disclosed
WO-2001081332-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2001-11-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020183362-A1 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation FPR2, FPR1, PTGES2 PTGS2 5/4885LMNA 4037/4885NPSR1 641/4885
US-20040092552-A1 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation FPR2, PTGES2, FPR1 PTGS2 5/4885LMNA 4107/4885NPSR1 618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.