SCHEMBL6723712

SCHEMBL6723712

Cc1csc2c1c(=O)[nH]c(=O)n2COCC[Si](C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 11/20 0.37
ERCC5 P28715 2/20 0.36
FEN1 P39748 2/20 0.36
PDE1B Q01064 2/20 0.34
ALDH1A1 P00352 1/20 0.33
PDE5A O76074 1/20 0.32
NPC1 O15118 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
PSMD14 O00487 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
EGLN1 Q9GZT9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6726529 0.81 ALDH1A1 (0.33) ALDH1A1PDE5ANPC1KDM4E
SCHEMBL6726785 0.72 NPC1 (0.37) ALDH1A1NPC1
SCHEMBL6719573 0.72 GRIK1 (0.47) ERCC5ALDH1A1PDE5ANPC1KDM4E
SCHEMBL25344514 0.71 ALDH1A1 (0.39) ALDH1A1NPC1KDM4EHPGDHTT
SCHEMBL6730106 0.71 ALDH1A1 (0.39) ALDH1A1NPC1
SCHEMBL25344264 0.71 TYMP (0.48) ALDH1A1HPGD
SCHEMBL6722438 0.70 ATM (0.38) ALDH1A1NPC1KDM4EMEN1HPGD
SCHEMBL6723898 0.68 PNP (0.36) ADORA2BALDH1A1NPC1MEN1HPGD
SCHEMBL6719104 0.68 NPC1 (0.53) ALDH1A1NPC1KDM4EMEN1HPGD
SCHEMBL6719388 0.68 MAPT (0.45) NPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673804-B1 PREVENTING OR TREATING ARTHRITIS (PARTICULARLY OSTEOARTHRITIS) OR INHIBITING METASTASIS, INVASION OR GROWTH OF CANCER (PARTICULARLY BREAST CANCER) SANKYO COMPANY, LIMITED (JP) 2004-01-06 US disclosed
EP-1069110-A1 SULFONAMIDE DERIVATIVES Sankyo Company Limited (JP) 2001-01-17 EP disclosed