SCHEMBL6726529

SCHEMBL6726529

Cc1csc2c(=O)[nH]c(=O)n(COCC[Si](C)(C)C)c12

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
PDE5A O76074 1/20 0.32
NPC1 O15118 1/20 0.32
KDM4E B2RXH2 1/20 0.31
PKM P14618 1/20 0.31
PDPK1 O15530 1/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
QPCT Q16769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6723712 0.81 ADORA2B (0.37) ALDH1A1PDE5ANPC1KDM4E
SCHEMBL6719573 0.77 GRIK1 (0.47) ALDH1A1PDE5ANPC1KDM4EPKM
SCHEMBL6726785 0.72 NPC1 (0.37) ALDH1A1NPC1
SCHEMBL25344514 0.71 ALDH1A1 (0.39) ALDH1A1NPC1KDM4EPKM
SCHEMBL6730106 0.71 ALDH1A1 (0.39) ALDH1A1NPC1
SCHEMBL25344264 0.71 TYMP (0.48) ALDH1A1
SCHEMBL6722438 0.70 ATM (0.38) ALDH1A1NPC1KDM4E
SCHEMBL6722467 0.69 PDE4A (0.60) ALDH1A1
SCHEMBL6719104 0.68 NPC1 (0.53) ALDH1A1NPC1KDM4ETNKSPARP1
SCHEMBL6723898 0.68 PNP (0.36) ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6673804-B1 PREVENTING OR TREATING ARTHRITIS (PARTICULARLY OSTEOARTHRITIS) OR INHIBITING METASTASIS, INVASION OR GROWTH OF CANCER (PARTICULARLY BREAST CANCER) SANKYO COMPANY, LIMITED (JP) 2004-01-06 US disclosed
EP-1069110-A1 SULFONAMIDE DERIVATIVES Sankyo Company Limited (JP) 2001-01-17 EP disclosed