SCHEMBL6741463

SCHEMBL6741463

[CH2]c1c(C)cc(N)cc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.47
TSHR P16473 5/20 0.47
PDE10A Q9Y233 1/20 0.40
CASP1 P29466 2/20 0.38
CYP3A4 P08684 6/20 0.36
TDP1 Q9NUW8 3/20 0.36
TP53 P04637 2/20 0.36
MAPK1 P28482 1/20 0.36
MAPT P10636 3/20 0.34
MEN1 O00255 2/20 0.34
THRB P10828 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ALOX15 P16050 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CD44 P16070 1/20 0.32
ACHE P22303 1/20 0.32
GAA P10253 2/20 0.31
NR4A1 P22736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylamine SCHEMBL27579793 0.75 RAPGEF4 (0.41) ALDH1A1TSHRTDP1TP53MAPT
SCHEMBL112391 0.73 ALDH1A1 (0.53) ALDH1A1TSHRPDE10ACASP1CYP3A4
SCHEMBL41001 0.73 RAPGEF4 (0.45) ALDH1A1TSHRTDP1TP53MAPT
SCHEMBL33589 0.73 ALDH1A1 (0.65) ALDH1A1TSHRPDE10ACASP1CYP3A4
SCHEMBL260795 0.73 ALDH1A1 (0.53) ALDH1A1TSHRPDE10ACASP1CYP3A4
SCHEMBL28040386 0.71 RAPGEF4 (0.43) ALDH1A1TSHRTDP1TP53MAPT
Hydrochloric Acid SCHEMBL23198661 0.71 ALDH1A1 (0.50) ALDH1A1TSHRPDE10ACASP1CYP3A4
Hydrochloric Acid SCHEMBL970560 0.71 ALDH1A1 (0.61) ALDH1A1TSHRPDE10ACASP1CYP3A4
Hydrochloric Acid SCHEMBL7931830 0.71 ALDH1A1 (0.61) ALDH1A1TSHRPDE10ACASP1CYP3A4
SCHEMBL3246567 0.71 ALDH1A1 (0.43) ALDH1A1TSHRPDE10ACASP1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689771-B2 TREATMENT OF RHEUMATOID ARTHRITIS, OSTEOARTHRITIS, PERIODONTITIS, GINGIVITIS, CORNEAL ULCERATION, SOLID TUMOR GROWTH BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-02-10 US disclosed
US-6376665-B1 ANTIARTHRITIC AGENTS, ANTIINFLAMMATORY AGENTS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2002-04-23 US disclosed