SCHEMBL6744349

SCHEMBL6744349

CCOC(=O)N1CSC[C@@H]1C(=O)N[C@@H](Cc1ccc(NC(=O)c2ccc(OC)cc2)cc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.46
CA2 P00918 1/20 0.44
ITGA4 P13612 6/20 0.44
ITGB1 P05556 5/20 0.44
NPC1 O15118 4/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
HIF1A Q16665 1/20 0.43
EPAS1 Q99814 1/20 0.43
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
EPHX2 P34913 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
POLB P06746 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6742904 0.93 ITGA4 (0.49) ITGA4ITGB1RAB9ASMN1; SMN2EPHX2
SCHEMBL6744943 0.92 ITGA4 (0.50) ITGA4ITGB1NPC1RAB9ASMN1; SMN2
SCHEMBL6742360 0.86 ITGB1 (0.46) FPR2ITGA4ITGB1KMT2A
SCHEMBL6741830 0.85 ITGA4 (0.54) ITGA4ITGB1NPC1ALDH1A1RAB9A
SCHEMBL6745542 0.84 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL6741663 0.84 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL27563993 0.83 ITGA4 (0.43) ITGA4ITGB1ALDH1A1
SCHEMBL6744273 0.83 ITGA4 (0.52) ITGA4ITGB1
SCHEMBL6745382 0.83 ITGA4 (0.39) CA2ITGA4ITGB1
SCHEMBL6741921 0.81 ITGB1 (0.47) ITGA4ITGB1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
CN-1313855-A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta UPJOHN CO (US) 2001-09-19 CN disclosed