SCHEMBL6744943

SCHEMBL6744943

CCOC(=O)N1CSC[C@@H]1C(=O)N[C@@H](Cc1ccc(NC(=O)c2ccccc2)cc1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 10/20 0.50
ITGB1 P05556 7/20 0.49
MMP9 P14780 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
RAB9A P51151 1/20 0.43
PREP P48147 1/20 0.42
ITGA5 P08648 1/20 0.42
CACNA1B Q00975 1/20 0.42
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
ITGA2B P08514 1/20 0.41
ITGB5 P18084 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6742904 0.94 ITGA4 (0.49) ITGA4ITGB1MMP9SMN1; SMN2GAA
SCHEMBL6741830 0.92 ITGA4 (0.54) ITGA4ITGB1SMN1; SMN2NPC1GAA
SCHEMBL6744349 0.92 FPR2 (0.46) ITGA4ITGB1SMN1; SMN2NPC1RAB9A
SCHEMBL6742360 0.89 ITGB1 (0.46) ITGA4ITGB1PREPITGA5CACNA1B
SCHEMBL6745542 0.88 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL6741663 0.88 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL6741921 0.87 ITGB1 (0.47) ITGA4ITGB1RAB9APREPITGA5
SCHEMBL6745377 0.87 ITGA4 (0.44) ITGA4ITGB1
SCHEMBL27563993 0.86 ITGA4 (0.43) ITGA4ITGB1PREPITGA5CACNA1B
SCHEMBL6744273 0.86 ITGA4 (0.52) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
CN-1313855-A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta UPJOHN CO (US) 2001-09-19 CN disclosed