SCHEMBL6741830

SCHEMBL6741830

CCOC(=O)N1CSC[C@@H]1C(=O)N[C@@H](Cc1ccc(NC(=O)c2cccnc2)cc1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 8/20 0.54
RAB9A P51151 5/20 0.47
NPC1 O15118 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
ITGAV P06756 2/20 0.45
ITGB3 P05106 1/20 0.45
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.44
POLB P06746 1/20 0.43
ITGB1 P05556 6/20 0.42
TP53 P04637 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
GFER P55789 1/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744943 0.92 ITGA4 (0.50) ITGA4RAB9ANPC1SMN1; SMN2ITGAV
SCHEMBL6742904 0.88 ITGA4 (0.49) ITGA4RAB9ASMN1; SMN2MAPTITGB1
SCHEMBL6744349 0.85 FPR2 (0.46) ITGA4RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL6742360 0.85 ITGB1 (0.46) ITGA4ITGAVITGB1MEN1KMT2A
SCHEMBL6741663 0.84 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL6745542 0.84 ITGA4 (0.57) ITGA4ITGB1
SCHEMBL27563993 0.82 ITGA4 (0.43) ITGA4ITGAVALDH1A1ITGB1
SCHEMBL6744273 0.82 ITGA4 (0.52) ITGA4ITGB1
SCHEMBL6741921 0.81 ITGB1 (0.47) ITGA4RAB9AITGAVMAPTITGB1
SCHEMBL6745377 0.81 ITGA4 (0.44) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
CN-1313855-A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta UPJOHN CO (US) 2001-09-19 CN disclosed