SCHEMBL6742360

SCHEMBL6742360

CCOC(=O)N1CSC[C@@H]1C(=O)N[C@@H](Cc1ccc(NC(C)=O)cc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.46
ITGA4 P13612 9/20 0.46
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PREP P48147 1/20 0.41
CACNA1B Q00975 1/20 0.40
ITGA5 P08648 3/20 0.40
ITGAV P06756 2/20 0.39
CYP2C19 P33261 1/20 0.39
FPR2 P25090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27563993 0.90 ITGA4 (0.43) ITGB1ITGA4PREPCACNA1BITGA5
SCHEMBL6744943 0.89 ITGA4 (0.50) ITGB1ITGA4PREPCACNA1BITGA5
SCHEMBL6742904 0.88 ITGA4 (0.49) ITGB1ITGA4
SCHEMBL6741921 0.87 ITGB1 (0.47) ITGB1ITGA4PREPCACNA1BITGA5
SCHEMBL6745542 0.86 ITGA4 (0.57) ITGB1ITGA4
SCHEMBL6741663 0.86 ITGA4 (0.57) ITGB1ITGA4
SCHEMBL6744349 0.86 FPR2 (0.46) ITGB1ITGA4KMT2AFPR2
SCHEMBL6742471 0.85 ITGA4 (0.52) ITGB1ITGA4
SCHEMBL6744273 0.85 ITGA4 (0.52) ITGB1ITGA4
SCHEMBL6741830 0.85 ITGA4 (0.54) ITGB1ITGA4MEN1KMT2AITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6685617-B1 4-(((-1-CARBOXY-2-(4-((2,6-DICHLOROBENZOYL)AMINE)PHENYL)ETHYL) AMINO)CARBONYL)-3-OXO-3-THIAZOLIDINEBUTANOIC ACID, USED AS ANTAGONISTS FOR CELLULAR ADHESION MOLECULES, AND ADMINISTERED AS ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY 2004-02-03 US disclosed
CN-1313855-A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta UPJOHN CO (US) 2001-09-19 CN disclosed