SCHEMBL6744930

SCHEMBL6744930

Cc1csc(-c2cccnc2-c2cc(F)c(S(N)(=O)=O)cc2F)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.39
PDE10A Q9Y233 1/20 0.39
CA1 P00915 5/20 0.36
CA2 P00918 5/20 0.36
ALOX5AP P20292 3/20 0.36
FEN1 P39748 3/20 0.36
PTGS2 P35354 3/20 0.36
CYP2E1 P05181 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2A6 P11509 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
MAPK1 P28482 1/20 0.34
CA9 Q16790 1/20 0.34
GLA P06280 1/20 0.34
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6718980 0.86 PTGS2 (0.43) TGFBR1PDE10ACA1CA2ALOX5AP
SCHEMBL6834803 0.84 CA1 (0.46) TGFBR1PDE10ACA1CA2PTGS2
SCHEMBL6749945 0.83 SCN9A (0.43) CA1CA2ALOX5APFEN1PTGS2
SCHEMBL6746037 0.83 ALOX5AP (0.44) CA1CA2ALOX5APFEN1PTGS2
SCHEMBL6746699 0.81 TGFBR1 (0.43) TGFBR1CA1CA2ALOX5APFEN1
SCHEMBL6750007 0.81 TGFBR1 (0.42) TGFBR1PDE10ACA1CA2ALOX5AP
SCHEMBL6744782 0.79 CA1 (0.39) CA1CA2ALOX5APFEN1PTGS2
SCHEMBL6749867 0.79 PTGS2 (0.49) CA1CA2ALOX5APFEN1PTGS2
SCHEMBL7042019 0.78 TGFBR1 (0.41) TGFBR1PDE10AALOX5APFEN1PTGS2
SCHEMBL6750040 0.77 PTGS2 (0.46) CA1CA2ALOX5APFEN1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US claimed
US-6699884-B2 ANTIINFLAMMATORY CYCLOOXYGENASE INHIBITORS. PHARMACIA CORPORATION 2004-03-02 US disclosed