SCHEMBL6745175

SCHEMBL6745175

N#Cc1c(F)cc(C=O)cc1F.N#Cc1c(F)cc(CO)cc1F

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.40
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2801373 0.86 TRPV4 (0.52) TRPV4CYP11B1CYP11B2PDCD1CD274
SCHEMBL2800490 0.86 TRPV4 (0.52) TRPV4EGFR
SCHEMBL28341814 0.77 TRPV4 (0.44) TRPV4CYP11B1CYP11B2PDCD1CD274
SCHEMBL7562408 0.75 CYP11B2 (0.47) TRPV4CYP11B1CYP11B2
SCHEMBL2726074 0.74 TRPV4 (0.48) TRPV4
SCHEMBL31371999 0.74 TRPV4 (0.39) TRPV4CYP11B1CYP11B2PDCD1CD274
SCHEMBL12465035 0.74 GRM5 (0.35) PDCD1CD274EGFR
SCHEMBL15157689 0.73 TRPV4 (0.40) TRPV4
SCHEMBL3839778 0.71 ACHE (0.42) EGFR
SCHEMBL13243340 0.71 ACHE (0.42) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1423362-A1 NEW MANDELIC ACID DERIVATIVES AND THEIR USE AS THROMBIN INHIBITORS AstraZeneca AB (SE) 2004-06-02 EP disclosed
WO-2003018551-A1 NEW MANDELIC ACID DERIVATIVES AND THEIR USE AS THROMBIN INHIBITORS ASTRAZENECA AB (SE) 2003-03-06 WO disclosed