SCHEMBL6750103

SCHEMBL6750103

CC1(C)OC[C@H](C[C@@H](Sc2cc(C(F)(F)F)cnc2C#N)c2ccccc2)N1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
FFAR4 Q5NUL3 1/20 0.32
RIPK1 Q13546 1/20 0.30
XIAP P98170 1/20 0.30
BIRC2 Q13490 1/20 0.30
TACR1 P25103 1/20 0.30
SCN10A Q9Y5Y9 1/20 0.30
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
LMNA P02545 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6750051 0.89 XIAP (0.30) ALDH1A1XIAPBIRC2HTT
SCHEMBL6746363 0.80 CYP2D6 (0.35) ALDH1A1XIAPBIRC2
SCHEMBL6751160 0.79 SMN1; SMN2 (0.32) SMN1; SMN2
SCHEMBL6750088 0.78 CYP2D6 (0.33) XIAPBIRC2
SCHEMBL6746343 0.77 CYP2D6 (0.33) ALDH1A1
SCHEMBL6750046 0.76 CYP2D6 (0.37) ALDH1A1
SCHEMBL4595258 0.76 ALDH1A1 (0.32) ALDH1A1HTT
SCHEMBL6750043 0.74 XIAP (0.32) ALDH1A1KMT2AXIAPBIRC2
SCHEMBL6750065 0.73 CYP2D6 (0.41) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL6752582 0.73 ITGB3 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040242871-A1 Novel arylheteroalkylamine derivatives ASTRAZENECA AB (SE) 2004-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040242871-A1 Novel arylheteroalkylamine derivatives CYP1A1, NOS3, NOS1 ALDH1A1 495/4885SMN1; SMN2 3507/4885MEN1 4748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.