SCHEMBL6761014

SCHEMBL6761014

N#C[CH]c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
ATM Q13315 1/20 0.42
NFE2L2 Q16236 7/20 0.42
HSD11B1 P28845 2/20 0.38
PKM P14618 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
APP P05067 1/20 0.37
PTGS1 P23219 1/20 0.37
FBP1 P09467 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7865937 0.76 RECQL (0.45) ALDH1A1MAPTMEN1KMT2A
SCHEMBL2986380 0.75 KDM4E (0.55) ALDH1A1GAAMAPTHTTATM
SCHEMBL18160982 0.75 KDM4E (0.55) ALDH1A1GAAMAPTHTTATM
SCHEMBL2986381 0.75 KDM4E (0.55) ALDH1A1GAAMAPTHTTATM
SCHEMBL18160977 0.75 KDM4E (0.55) ALDH1A1GAAMAPTHTTATM
SCHEMBL22065499 0.75 KDM4E (0.55) ALDH1A1GAAMAPTHTTATM
SCHEMBL9512577 0.74 ALDH1A1 (0.46) ALDH1A1MAPTNFE2L2L3MBTL1PTGS1
SCHEMBL7867492 0.74 ALDH1A1 (0.47) ALDH1A1GAAMAPTL3MBTL1FBP1
SCHEMBL3227313 0.74 NFE2L2 (0.42) NFE2L2HSD11B1APPPTGS1FBP1
SCHEMBL3981306 0.74 HSD17B10 (0.46) GAAFBP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743790-B2 A UREA OR THIOUREA DERIVATIVES CONTAINING AMIDE GROUP USEFUL AS ANTICOAGULANTS AND ANTIINFLAMMATORY AGENTS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-06-01 US disclosed
EP-1299354-A2 FACTOR VIIA INHIBITORY (THIO)UREA DERIVATIVES, THEIR PREPARATION AND THEIR USE Aventis Pharma Deutschland GmbH (DE) 2003-04-09 EP disclosed
WO-2001094301-A2 FACTOR VIIA INHIBITORY (THIO)UREA DERIVATIVES, THEIR PREPARATION AND THEIR USE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-12-13 WO disclosed
EP-1162194-A1 Factor VIIa inhibitory (thio)urea derivatives, their preparation and their use Aventis Pharma Deutschland GmbH (DE) 2001-12-12 EP disclosed
EP-0253536-A2 Fluorobenzyl esters IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-01-20 EP disclosed