SCHEMBL6765071

SCHEMBL6765071

NS(=O)(=O)c1ccc(C(=O)N2Cc3ccc(C#CCc4ccc(Cl)cc4)cc3C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA1 P00915 20/20 0.53
CA2 P00918 20/20 0.53
CA9 Q16790 20/20 0.53
CA7 P43166 15/20 0.53
CA14 Q9ULX7 15/20 0.53
CA12 O43570 15/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6765068 0.75 MMP13 (0.45) CA1CA2CA9CA7CA14
SCHEMBL5697123 0.72 MMP13 (0.42) CA1CA2CA9CA7CA14
SCHEMBL6761897 0.71 ACACB (0.44)
SCHEMBL16053390 0.65 CA1 (0.70) CA1CA2CA9CA7CA14
SCHEMBL21768167 0.65 MAOB (0.56) CA1CA2CA9CA7CA14
SCHEMBL30089453 0.65 MAOB (0.56) CA1CA2CA9CA7CA14
SCHEMBL14493373 0.64 CA12 (0.87) CA1CA2CA9CA7CA14
SCHEMBL6705933 0.63 POLB (0.39)
SCHEMBL23628467 0.62 CA1 (0.63) CA1CA2CA9CA7CA14
SCHEMBL14157570 0.62 CA1 (0.50) CA1CA2CA9CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040038973-A1 Treating osteoarthritis or rheumatoid arthritis NAHRA JOE (US) 2004-02-26 US claimed
WO-2004014365-A1 PHTHALIMIDE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed
US-20040038973-A1 Treating osteoarthritis or rheumatoid arthritis NAHRA JOE (US) 2004-02-26 US disclosed
WO-2004014365-A1 PHTHALIMIDE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040038973-A1 Treating osteoarthritis or rheumatoid arthritis MMP13, MMP11, MMP9 CA1 724/4885CA2 300/4885CA9 279/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.