SCHEMBL6766920

SCHEMBL6766920

O=C1COC(c2ccccc2O)=NN1c1ccccc1Br

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.53
MAOB P27338 3/20 0.40
MGLL Q99685 1/20 0.33
HSP90AA1 P07900 1/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TSHR P16473 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TP53 P04637 1/20 0.31
EP300 Q09472 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6768472 0.86 CYP2D6 (0.51) CYP2D6MAOBMGLLHSP90AA1ALDH1A1
SCHEMBL6766055 0.81 CASP6 (0.41) CYP2D6MAOBALDH1A1HPGDL3MBTL1
SCHEMBL6763490 0.81 CYP2D6 (0.54) CYP2D6MAOBHSP90AA1SMN1; SMN2TSHR
SCHEMBL5780097 0.81 KMT2A (0.37) CYP2D6MAOBMGLLTSHRKMT2A
SCHEMBL6766363 0.78 CYP2D6 (0.47) CYP2D6MAOBALDH1A1MEN1KMT2A
SCHEMBL10633526 0.77 KMT2A (0.50) MAOBNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL5780049 0.77 SLC5A2 (0.36) CYP2D6MGLLNPC1RAB9ASMN1; SMN2
SCHEMBL6763578 0.77 CYP2D6 (0.50) CYP2D6MAOBNPC1RAB9AALDH1A1
SCHEMBL6766166 0.76 CYP2D6 (0.40) CYP2D6MAOBALDH1A1HPGDMEN1
SCHEMBL5781166 0.75 HTR7 (0.46) MAOBRAB9ASMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP claimed
US-6825192-B1 NON-N-METHYL-D-ASPARTATE (NON- NMDA) EXCITATORY AMINO ACID RECEPTOR ANTAGONISTIC ACTION, FOR EXAMPLE 2-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) RECEPTOR ANTAGONISTIC ACTION EISAI CO., LTD. (JP) 2004-11-30 US disclosed
EP-1153922-A1 HETERODIAZINONE DERIVATIVES Eisai Co., Ltd. (JP) 2001-11-14 EP disclosed