SCHEMBL6767276

SCHEMBL6767276

Fc1cc(F)cc(C[CH]c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.40
AHR P35869 1/20 0.40
NQO2 P16083 1/20 0.39
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37
CYP1A2 P05177 1/20 0.37
BACE1 P56817 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
IDO1 P14902 2/20 0.35
FBP1 P09467 1/20 0.35
MAOB P27338 2/20 0.35
HIF1A Q16665 1/20 0.35
EPAS1 Q99814 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790207 0.83 TAAR1 (0.47) PTGS1AHRNQO2CYP1A2TAAR1
SCHEMBL8366212 0.80 IDO1 (0.39) PTGS1BACE1IDO1
SCHEMBL4811925 0.78 ALDH1A1 (0.48) CYP1A1CYP1B1BACE1MAOB
SCHEMBL5323954 0.77 TAAR1 (0.50) TAAR1IDO1MAOB
SCHEMBL3590959 0.76 TAAR1 (0.44) PTGS1AHRNQO2TAAR1IDO1
SCHEMBL28757558 0.74 ALDH1A1 (0.48) CYP1A1CYP1B1TAAR1IDO1MAOB
SCHEMBL1992348 0.70 PTGS1 (0.46) PTGS1AHRNQO2CYP1A1CYP1B1
SCHEMBL1295918 0.68 RXRA (0.41) IDO1
SCHEMBL16225102 0.68 LMNA (0.44) PTGS1CYP1A2
SCHEMBL14396108 0.68 IDO1 (0.39) CLK1DYRK1AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787540-B2 FOR THERAPY OF AUTOIMMUNE DISEASES, ASTHMA, OSTEOPOROSIS, ATHEROSCLEROSIS, ALZHEIMER'S DISEASE BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2004-09-07 US disclosed