SCHEMBL6770869

SCHEMBL6770869

O=C(c1ccc(F)c([N+](=O)[O-])c1)c1ccccn1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B14 Q9BPX1 1/20 0.64
ITGB1 P05556 1/20 0.53
ITGA5 P08648 1/20 0.53
AURKB Q96GD4 1/20 0.52
KMT2A Q03164 5/20 0.50
ALDH1A1 P00352 3/20 0.49
MEN1 O00255 4/20 0.48
MAPT P10636 3/20 0.48
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
IRAK4 Q9NWZ3 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
HTT P42858 2/20 0.45
LMNA P02545 2/20 0.45
VCAM1 P19320 2/20 0.45
KDM4E B2RXH2 2/20 0.44
GMNN O75496 1/20 0.44
TTR P02766 1/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11880101 0.85 AURKB (0.70) HSD17B14AURKBKMT2AALDH1A1MEN1
SCHEMBL9383490 0.84 MAPT (0.66) HSD17B14AURKBKMT2AALDH1A1MEN1
SCHEMBL11715543 0.84 LMNA (0.56) HSD17B14AURKBKMT2AALDH1A1MEN1
Bromide SCHEMBL11874976 0.84 AURKB (0.68) HSD17B14AURKBKMT2AALDH1A1MEN1
SCHEMBL7363433 0.81 TTR (0.60) HSD17B14AURKBKMT2AALDH1A1MEN1
SCHEMBL4605109 0.81 VCAM1 (0.62) ITGB1ITGA5KMT2AALDH1A1MEN1
SCHEMBL11875218 0.81 RAB9A (0.69) AURKBKMT2AALDH1A1MEN1MAPT
Methyl Alcohol SCHEMBL28111073 0.80 VCAM1 (0.64) ITGB1ITGA5KMT2AALDH1A1MEN1
Bromide SCHEMBL7367632 0.80 TTR (0.59) HSD17B14AURKBKMT2AALDH1A1MEN1
SCHEMBL7497537 0.80 VCAM1 (0.68) ITGB1ITGA5KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6706663-B2 CHEMICAL INTERMEDIATES WYETH 2004-03-16 US disclosed
US-20020028748-A1 Herbicidal 3 -heterocyclic substituted benzisothiazole and benzisoxazole compounds INTELLECTUAL PROPERTY DEPARTMENT BASF AKTIENGESELLSCHAFT (DE) 2002-03-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020028748-A1 Herbicidal 3 -heterocyclic substituted benzisothiazole and benzisoxazole compounds CYP4X1, HAX1, DDT HSD17B14 2205/4885ITGB1 4299/4885ITGA5 4662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.