SCHEMBL6771848

SCHEMBL6771848

CCC(C)Cc1ccc(Br)cc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.41
ACACB O00763 1/20 0.40
PYCR1 P32322 1/20 0.39
TAAR1 Q96RJ0 3/20 0.39
KMT2A Q03164 2/20 0.39
MME P08473 3/20 0.38
HTR2A P28223 1/20 0.38
EPHX1 P07099 1/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8687580 0.94 SIGMAR1 (0.41) SIGMAR1ACACBPYCR1TAAR1KMT2A
SCHEMBL8687584 0.94 SIGMAR1 (0.41) SIGMAR1ACACBPYCR1TAAR1KMT2A
SCHEMBL15161169 0.81 TP53 (0.42) ACACBTAAR1
SCHEMBL9026591 0.80 ACACB (0.42) SIGMAR1ACACBPYCR1TAAR1KMT2A
SCHEMBL10041 0.80 ACACB (0.42) SIGMAR1ACACBPYCR1TAAR1KMT2A
SCHEMBL9284510 0.80 ACACB (0.42) SIGMAR1ACACBPYCR1TAAR1KMT2A
SCHEMBL17393790 0.80 TAAR1 (0.46) SIGMAR1ACACBPYCR1TAAR1HTR2A
SCHEMBL10823884 0.80 SIGMAR1 (0.40) SIGMAR1ACACBPYCR1TAAR1KMT2A
SCHEMBL28734578 0.79 SLC6A4 (0.39) TAAR1
SCHEMBL5838111 0.79 IDO1 (0.42) ACACBTAAR1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8772507-B2 Imidazole-benzamide anti-cancer agents CYTOKINETICS, INC. (US) 2014-07-08 US disclosed
US-20130096315-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS QIAN XIANGPING (US) 2013-04-18 US disclosed
US-20120283287-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS QIAN XIANGPING (US) 2012-11-08 US disclosed
WO-2010149684-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-29 WO disclosed
US-6673824-B1 HYPOTENSIVE AGENTS BRISTOL-MYERS SQUIBB CO. 2004-01-06 US disclosed
US-6107320-A Phenyl sulfonamide endothelin antagonists BRISTOL-MYERS SQUIBB CO. (US) 2000-08-22 US disclosed
US-5514696-A Phenyl sulfonamide endothelin antagonists BRISTOL-MYERS SQUIBB CO. (US) 1996-05-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120283287-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS KIF5B, KIF2C, PLK1 SIGMAR1 3812/4885ACACB 903/4885PYCR1 2760/4885
US-20130096315-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS KIF5B, KIF2C, PLK1 SIGMAR1 3721/4885ACACB 621/4885PYCR1 2886/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.