SCHEMBL677185

SCHEMBL677185

Cc1ccc(C(=O)OB(O)O)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.59
ALDH1A1 P00352 7/20 0.50
LMNA P02545 2/20 0.50
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
SMN1; SMN2 Q16637 3/20 0.48
MAPT P10636 2/20 0.47
PKM P14618 2/20 0.45
HTT P42858 2/20 0.45
ATM Q13315 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
HPGD P15428 1/20 0.45
NLRP1 Q9C000 1/20 0.45
GAA P10253 1/20 0.45
MEN1 O00255 1/20 0.45
NTSR1 P30989 1/20 0.45
KMT2A Q03164 1/20 0.45
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
NPC1 O15118 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16897249 0.84 TDP1 (0.61) TDP1ALDH1A1LMNACES2CES1
SCHEMBL15971711 0.80 TSHR (0.55) ALDH1A1CES2CES1SMN1; SMN2MAPT
SCHEMBL16897300 0.78 CES2 (0.50) CES2CES1SMN1; SMN2MAPTPKM
SCHEMBL28628636 0.78 LMNA (0.52) TDP1ALDH1A1LMNAMAPTPKM
SCHEMBL11228311 0.77 LMNA (0.58) TDP1ALDH1A1LMNACES2CES1
SCHEMBL248492 0.77 TDP1 (0.70) TDP1ALDH1A1LMNACES2CES1
SCHEMBL6654554 0.77 TDP1 (0.70) TDP1ALDH1A1LMNACES2CES1
SCHEMBL64626 0.77 TDP1 (0.70) TDP1ALDH1A1LMNACES2CES1
SCHEMBL9860907 0.76 LMNA (0.56) TDP1ALDH1A1LMNACES2CES1
Ammonia Solution, Strong SCHEMBL8998037 0.76 LMNA (0.56) TDP1ALDH1A1LMNACES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944750-B2 Polyethylene glycol substituted acyl borates ETH ZURICH (CH) 2018-04-17 US disclosed
EP-3092263-B1 POLYETHYLENE GLYCOL SUBSTITUTED ACYL BORATES ETH ZUERICH (CH) 2018-02-21 EP disclosed
US-20170022321-A1 POLYETHYLENE GLYCOL SUBSTITUTED ACYL BORATES ETH ZURICH (CH) 2017-01-26 US disclosed
EP-3092263-A1 POLYETHYLENE GLYCOL SUBSTITUTED ACYL BORATES ETH Zurich (CH) 2016-11-16 EP disclosed
WO-2015104374-A1 POLYETHYLENE GLYCOL SUBSTITUTED ACYL BORATES ETH ZURICH (CH) 2015-07-16 WO disclosed
US-8283401-B2 Conjugated diene polymer manufacturing method, polybutadiene, and rubber composition utilizing the same UBE INDUSTRIES, LTD (JP) 2012-10-09 US disclosed
US-20110269899-A1 CONJUGATED DIENE POLYMER MANUFACTURING METHOD, POLYBUTADIENE, AND RUBBER COMPOSITION UTILIZING THE SAME UBE INDUSTRIES, LTD. (JP) 2011-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170022321-A1 POLYETHYLENE GLYCOL SUBSTITUTED ACYL BORATES BRS3, FFAR3, LPAR3 TDP1 4349/4885ALDH1A1 3912/4885LMNA 1255/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.