SCHEMBL6771955

SCHEMBL6771955

CC(C)(C)c1nn(-c2ccc(I)cc2)c2c1C(=O)CCC2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.41
SRC P12931 1/20 0.39
GRIA2 P42262 10/20 0.38
CYP1A2 P05177 4/20 0.38
CYP2C9 P11712 4/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
GAA P10253 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6167303 0.86 ALDH1A1 (0.45) OPRM1SRCHTTKDM4EALDH1A1
SCHEMBL6770286 0.83 OPRM1 (0.56) OPRM1SRCHTTKDM4EALDH1A1
SCHEMBL6766781 0.80 OPRM1 (0.54) OPRM1SRC
SCHEMBL6771234 0.80 CSNK2A2 (0.35) OPRM1HTTALDH1A1
SCHEMBL6767074 0.79 OPRM1 (0.41) OPRM1SRCGRIA2CYP1A2CYP2C9
SCHEMBL6767118 0.79 HTT (0.40) OPRM1SRCGRIA2HTTKDM4E
SCHEMBL6772487 0.79 SRC (0.53) OPRM1SRCHTTKDM4EALDH1A1
SCHEMBL6766716 0.78 HTT (0.37) OPRM1SRCGRIA2HTTALDH1A1
SCHEMBL6771178 0.77 SRC (0.43) OPRM1SRCGRIA2HTTKDM4E
SCHEMBL6776541 0.77 ALDH1A1 (0.47) OPRM1SRCCYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed