SCHEMBL6776541

SCHEMBL6776541

CCCc1nn(-c2ccc(I)cc2)c2c1C(=O)CCC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
MAPT P10636 1/20 0.47
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
TSHR P16473 1/20 0.43
OPRM1 P35372 4/20 0.39
SRC P12931 2/20 0.38
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
ALPL P05186 1/20 0.35
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6162867 0.87 ALDH1A1 (0.49) ALDH1A1MAPTLMNAHTTTSHR
SCHEMBL6770454 0.85 ALDH1A1 (0.48) ALDH1A1MAPTLMNAHTTTSHR
SCHEMBL6767118 0.84 HTT (0.40) ALDH1A1MAPTLMNAHTTTSHR
SCHEMBL6770286 0.81 OPRM1 (0.56) ALDH1A1HTTTSHROPRM1SRC
SCHEMBL6767582 0.81 ALDH1A1 (0.56) ALDH1A1LMNAOPRM1KMT2ANPSR1
SCHEMBL6771081 0.80 ALDH1A1 (0.58) ALDH1A1MAPTLMNAHTTTSHR
SCHEMBL6766716 0.78 HTT (0.37) ALDH1A1MAPTLMNAHTTTSHR
SCHEMBL6777584 0.78 ALDH1A1 (0.53) ALDH1A1MAPTLMNAHTTTSHR
SCHEMBL6767248 0.78 DHODH (0.35) ALDH1A1MAPTLMNAKMT2ANPSR1
SCHEMBL6771955 0.77 OPRM1 (0.41) ALDH1A1HTTOPRM1SRCKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed