SCHEMBL6772135

SCHEMBL6772135

COc1ccc(CNC(=O)C2(CCCCBr)c3ccccc3-c3ccccc32)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.49
GAA P10253 2/20 0.47
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
PKM P14618 1/20 0.45
CYP2C19 P33261 1/20 0.45
RECQL P46063 1/20 0.45
HSD17B10 Q99714 1/20 0.45
EPHX2 P34913 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771541 0.86 MMP13 (0.50) ALDH1A1SMN1; SMN2EPHX2
SCHEMBL6770262 0.86 NPC1 (0.48) ALDH1A1MEN1KMT2A
SCHEMBL6771867 0.85 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL7600342 0.85 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2GAAMEN1KMT2A
SCHEMBL5863883 0.83 SMN1; SMN2 (0.42) SMN1; SMN2
SCHEMBL6771247 0.82 TAS1R3 (0.51) ALDH1A1GAAMEN1KMT2APKM
SCHEMBL6766560 0.80 POLB (0.45) ALDH1A1MEN1KMT2ARECQL
SCHEMBL6771422 0.79 HTT (0.44) ALDH1A1SMN1; SMN2GAA
SCHEMBL6771465 0.78 MTTP (0.47)
SCHEMBL6770628 0.77 MTTP (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6821967-B2 AMINES SUCH AS 9-(4-(4-(BENZOTHIAZOL-2-YL)-PIPERAZIN-1-YL)-BUTYL)-9H-FLUORENE-9-CARBOXYLIC ACID (2,2,2-TRIFLUOROETHYL) AMIDE, USED AS MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN ANTAGONISTS, TO PREVENT ATHEROSCLEROSIS OR HYPERLIPEMIA BOEHRINGER INGELHEIM PHARMA KG (DE) 2004-11-23 US disclosed
US-20030166637-A1 Substituted piperazine derivatives, the preparation thereofand their use as medicaments BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030166637-A1 Substituted piperazine derivatives, the preparation thereofand their use as medicaments MTTP, CETP, CPT1A ALDH1A1 715/4885SMN1; SMN2 4276/4885GAA 1187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.