SCHEMBL7600342

SCHEMBL7600342

COc1ccc(CNC(=O)OC2(CCCCBr)c3ccccc3-c3ccccc32)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 1/20 0.47
GAA P10253 2/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
PKM P14618 1/20 0.43
CYP2C19 P33261 1/20 0.43
EPHX2 P34913 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
POLB P06746 1/20 0.42
NOD2 Q9HC29 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599607 0.87 NPC1 (0.46) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL7596015 0.86 MMP13 (0.48) ALDH1A1SMN1; SMN2GAAMEN1KMT2A
SCHEMBL7596021 0.85 HDAC1 (0.45) ALDH1A1GAAMEN1KMT2A
SCHEMBL6772135 0.85 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2GAAMEN1KMT2A
SCHEMBL7599929 0.84 TP53 (0.39) SMN1; SMN2GAAMEN1KMT2AEPHX2
SCHEMBL7593148 0.84 PDK2 (0.40)
SCHEMBL7594799 0.82 TAS1R3 (0.49) ALDH1A1GAAMEN1KMT2APKM
SCHEMBL7596505 0.82 POLB (0.41) ALDH1A1SMN1; SMN2GAAMEN1KMT2A
SCHEMBL7596777 0.80 HTT (0.41) ALDH1A1SMN1; SMN2GAACYP3A4POLB
SCHEMBL7600206 0.79 PDK2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255736-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) Boehringer Ingelheim Pharma KG (DE) 2002-11-13 EP disclosed
WO-2001047898-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed