SCHEMBL6773336

SCHEMBL6773336

CCOC(=O)NCc1ccc2[nH]c(=O)[nH]c2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
KDM4E B2RXH2 4/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
ALDH1A1 P00352 7/20 0.47
MAPT P10636 5/20 0.47
GAA P10253 3/20 0.47
ALOX15 P16050 2/20 0.47
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PKM P14618 1/20 0.45
POLB P06746 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6763547 0.87 TSHR (0.56) TSHRSMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL10209975 0.82 L3MBTL1 (0.47) SMN1; SMN2KDM4EALDH1A1MAPTGAA
SCHEMBL6763567 0.78 SMN1; SMN2 (0.54) SMN1; SMN2ALDH1A1MAPTGAAALOX15
SCHEMBL10599026 0.78 TSHR (0.70) TSHRSMN1; SMN2KDM4ECYP1A2CYP3A4
SCHEMBL13415005 0.77 TSHR (0.57) TSHRSMN1; SMN2KDM4ECYP1A2CYP3A4
SCHEMBL6767362 0.76 PDE3B (0.65) SMN1; SMN2KDM4EALDH1A1MAPTGAA
SCHEMBL7788580 0.76 TSHR (0.67) TSHRSMN1; SMN2KDM4ECYP1A2CYP3A4
SCHEMBL6768232 0.74 GAA (0.47) KDM4EALDH1A1MAPTGAAALOX15
SCHEMBL12332829 0.74 GAA (0.54) SMN1; SMN2KDM4EALDH1A1MAPTGAA
SCHEMBL6768134 0.74 NLRP3 (0.41) TSHRSMN1; SMN2KDM4ECYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6699880-B1 STIMULATE MUSCARINIC ACETYLCHOLINE RECEPTORS M4, ANALGESICS BANYU PHARMACEUTICAL CO., LTD. (JP) 2004-03-02 US disclosed
EP-1221443-A1 SUBSTITUTED IMIDAZOLIDINONE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 2002-07-10 EP disclosed