SCHEMBL6775235

SCHEMBL6775235

CN(C)C(=O)c1ccc(N(CCCOc2ccc3ccnc(N)c3c2)C(=O)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.36
F10 P00742 2/20 0.34
PDE10A Q9Y233 1/20 0.34
PDK2 Q15119 3/20 0.33
PDK4 Q16654 3/20 0.33
MAOB P27338 1/20 0.33
AOC3 Q16853 1/20 0.33
THRA P10827 1/20 0.33
GPR119 Q8TDV5 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
HCRTR2 O43614 1/20 0.32
ALDH1A1 P00352 2/20 0.32
USP2 O75604 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6770185 0.95 TBXAS1 (0.36) TBXAS1F10PDK2PDK4MAOB
SCHEMBL6769131 0.84 HRH3 (0.43) F10MAOBAOC3HRH3ALDH1A1
SCHEMBL6890251 0.83 F10 (0.38) F10ALDH1A1LMNACNR2
Trifluoroacetic Acid SCHEMBL6775232 0.80 RAD52 (0.42) F10ALDH1A1
SCHEMBL6765996 0.80 HRH3 (0.41) F10MAOBAOC3HRH3ALDH1A1
Trifluoroacetic Acid SCHEMBL6770182 0.79 NPC1 (0.42) F10ALDH1A1HPGDSMN1; SMN2
SCHEMBL3911248 0.73 F10 (0.50) F10
Trifluoroacetic Acid SCHEMBL6775993 0.71 F10 (0.42) F10ALDH1A1HPGDSMN1; SMN2
SCHEMBL6775981 0.69 KDM4E (0.40) F10ALDH1A1
SCHEMBL6769241 0.68 ROCK1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825181-B1 ORALLY ADMINISTRATED TO EXHIBIT A STRONG ANTICOAGULANT EFFECT BY INHIBITING ACTIVATED BLOOD- COAGULATION FACTOR X AJINOMOTO CO., INC. (JP) 2004-11-30 US disclosed
EP-1065200-A1 AMINOISOQUINOLINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2001-01-03 EP disclosed