SCHEMBL6769241

SCHEMBL6769241

Nc1nccc2ccc(OCCCNC(=O)O)cc12

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.45
MTNR1A P48039 17/20 0.43
MTNR1B P49286 16/20 0.43
PLAU P00749 1/20 0.40
PLAT P00750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6776349 0.96 ROCK1 (0.46) ROCK1MTNR1AMTNR1BPLAUPLAT
Trifluoroacetic Acid SCHEMBL6775232 0.78 RAD52 (0.42)
SCHEMBL6769265 0.78 PLAU (0.43) ROCK1MTNR1AMTNR1BPLAUPLAT
SCHEMBL7120850 0.77 ROCK1 (0.45) ROCK1PLAUPLAT
Trifluoroacetic Acid SCHEMBL6769129 0.76 F10 (0.53)
Trifluoroacetic Acid SCHEMBL6890249 0.76 F10 (0.49) ROCK1MTNR1AMTNR1B
SCHEMBL6775414 0.76 ROCK1 (0.41) ROCK1PLAU
SCHEMBL6982099 0.76 F12 (0.44) ROCK1PLAUPLAT
SCHEMBL20982809 0.76 L3MBTL1 (0.46) MTNR1AMTNR1B
Trifluoroacetic Acid SCHEMBL6770182 0.75 NPC1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825181-B1 ORALLY ADMINISTRATED TO EXHIBIT A STRONG ANTICOAGULANT EFFECT BY INHIBITING ACTIVATED BLOOD- COAGULATION FACTOR X AJINOMOTO CO., INC. (JP) 2004-11-30 US disclosed
EP-1065200-A1 AMINOISOQUINOLINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2001-01-03 EP disclosed