SCHEMBL6775893

SCHEMBL6775893

O=C1[C@@H]2CC[C@H](CN1CCCc1ccccc1)N2Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.49
HRH3 Q9Y5N1 1/20 0.44
OPRD1 P41143 3/20 0.44
OPRK1 P41145 2/20 0.44
SIGMAR1 Q99720 6/20 0.42
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
FAAH O00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6781973 0.96 SIGMAR1 (0.46) OPRM1HRH3OPRD1OPRK1SIGMAR1
SCHEMBL6775421 0.89 OPRM1 (0.40) OPRM1HRH3SIGMAR1
SCHEMBL6784683 0.85 OPRM1 (0.41) OPRM1HRH3OPRD1OPRK1SIGMAR1
SCHEMBL6779579 0.85 BCHE (0.42) OPRM1SIGMAR1
SCHEMBL6784327 0.82 SIGMAR1 (0.47) SIGMAR1
SCHEMBL6779637 0.79 CHRNB2 (0.39) OPRM1OPRK1
SCHEMBL6779144 0.78 SIGMAR1 (0.50) SIGMAR1
SCHEMBL6780693 0.77 SIGMAR1 (0.42) OPRM1HRH3SIGMAR1
SCHEMBL6774415 0.75 BCHE (0.39) OPRM1SIGMAR1
SCHEMBL14410729 0.74 CHRM2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed