SCHEMBL6780693

SCHEMBL6780693

O=C1[C@@H]2CC[C@H](CN1C(CCc1ccccc1)CCc1ccccc1)N2Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.42
HRH3 Q9Y5N1 1/20 0.41
OPRM1 P35372 1/20 0.39
ALDH1A1 P00352 2/20 0.38
ACE P12821 2/20 0.37
ALKBH5 Q6P6C2 1/20 0.36
CHRM2 P08172 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRM3 P20309 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
S1PR1 P21453 1/20 0.35
S1PR5 Q9H228 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6779167 0.81 SIGMAR1 (0.46) SIGMAR1ALDH1A1CHRM3CHRM5
SCHEMBL6775893 0.77 OPRM1 (0.49) SIGMAR1HRH3OPRM1
SCHEMBL6781973 0.76 SIGMAR1 (0.46) SIGMAR1HRH3OPRM1
SCHEMBL6784683 0.76 OPRM1 (0.41) SIGMAR1HRH3OPRM1ALDH1A1ACE
SCHEMBL6775421 0.71 OPRM1 (0.40) SIGMAR1HRH3OPRM1ALDH1A1ALKBH5
SCHEMBL10008035 0.70 ALDH1A1 (0.62) ALDH1A1MEN1KMT2ANPSR1
SCHEMBL6949097 0.69 SIGMAR1 (0.49) SIGMAR1HRH3ALDH1A1ALKBH5CHRM2
Hydrochloric Acid SCHEMBL5965726 0.68 ALDH1A1 (0.60) ALDH1A1CHRM2MEN1KMT2ACHRM4
SCHEMBL11776863 0.68 ALDH1A1 (0.47) HRH3ALDH1A1CHRM2MEN1KMT2A
SCHEMBL21308106 0.67 SIGMAR1 (0.44) SIGMAR1HRH3ALDH1A1ALKBH5CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6818643-B1 3,9-DIAZABICYCLO(3.3.1)NONAN-2-ONE DERIVATIVES; PEPTIDYL-PROLYL ISOMERASE (PPIASE OR ROTAMASE) INHIBITORS; NEUROPROTECTIVE AGENTS BRISTOL-MYERS SQUIBB COMPANY 2004-11-16 US disclosed