SCHEMBL6790733

SCHEMBL6790733

CC1CN(c2ccc3cc[nH]c3c2)CC(C)N1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.43
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
AHR P35869 3/20 0.40
CMA1 P23946 1/20 0.40
TYR P14679 1/20 0.40
KCNH2 Q12809 4/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
MAPT P10636 1/20 0.37
ALOX12 P18054 1/20 0.37
ENPP2 Q13822 2/20 0.37
CYP2A6 P11509 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6840540 0.89 KCNH2 (0.46) AHRKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL17542571 0.83 MAPT (0.44) GHSRMEN1POLBMAPK1KMT2A
SCHEMBL20157184 0.76 MAPT (0.46) GHSRMEN1POLBMAPK1KMT2A
SCHEMBL6783725 0.76 TGFBR1 (0.38) GHSRMEN1POLBKMT2AKCNH2
SCHEMBL5097444 0.76 HTR3A (0.57) MEN1POLBMAPK1KMT2AKDM4E
SCHEMBL3342144 0.73 TERT (0.52) MEN1POLBMAPK1KMT2AAHR
SCHEMBL21388458 0.71 ADRB1 (0.49) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL5382950 0.71 TERT (0.53) MEN1POLBMAPK1KMT2AAHR
SCHEMBL9983829 0.71 AR (0.48) GHSRAHRCMA1TYRKDM4E
SCHEMBL23072821 0.70 MAPT (0.41) GHSRMEN1MAPK1KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6747030-B1 CIS-6-(3,5-DIMETHYLPIPERAZIN-1-YL)-5-METHOXY-1-(2'-METHYL-4'-( 5-METHYL-1,2,4-OXADIAZOL-3-YL)BIPHENYL-4-CARBONYL)INDOLINE, ITS HYDROCHLORIDE SALT, OR ANOTHER PHARMACEUTICALLY ACCEPTABLE SALT THEREOF; ANTIDEPRESSANTS SMITHKLINE BEECHAM P.L.C. (GB) 2004-06-08 US disclosed