SCHEMBL6790843

SCHEMBL6790843

COc1ccc(CCNC(=O)c2ccc(C(=O)O)s2)cc1OC

nearest known ligand 0.78

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.78
LMNA P02545 2/20 0.78
GAA P10253 2/20 0.59
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA9 Q16790 1/20 0.59
KMT2A Q03164 2/20 0.58
ALDH1A1 P00352 2/20 0.57
POLB P06746 1/20 0.56
MAPT P10636 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9408887 0.81 NAMPT (0.67) NAMPTLMNAGAACA12CA1
SCHEMBL901614 0.80 CA12 (0.73) NAMPTLMNAGAACA12CA1
SCHEMBL29356619 0.79 ALDH1A1 (0.77) NAMPTGAACA1CA2CA9
SCHEMBL6270935 0.79 ALDH1A1 (0.77) NAMPTGAACA1CA2CA9
SCHEMBL27888928 0.79 NAMPT (1.00) NAMPTLMNAGAAKMT2AALDH1A1
SCHEMBL7274134 0.77 NPC1 (0.85) LMNAGAACA1CA2CA9
SCHEMBL8099685 0.77 CA1 (0.73) LMNAGAACA12CA1CA2
SCHEMBL10359474 0.77 CA12 (0.73) NAMPTGAACA12CA1CA2
SCHEMBL2224069 0.77 CA12 (0.73) GAACA12CA1CA2CA9
SCHEMBL7265002 0.77 CA12 (0.73) NAMPTLMNAGAACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6784173-B2 ANTIPROLIFERATIVE AGENTS; ANTITUMOR AGENTS HOFFMANN-LA ROCHE INC. 2004-08-31 US claimed