SCHEMBL6796063

SCHEMBL6796063

CC(=O)N(C(C)=O)c1ncccc1C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 4/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 2/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
RAB9A P51151 3/20 0.44
MAPT P10636 3/20 0.44
NPC1 O15118 1/20 0.44
AHR P35869 1/20 0.44
HTT P42858 1/20 0.43
NAPRT Q6XQN6 2/20 0.41
P2RX7 Q99572 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
BLM P54132 1/20 0.38
AGER Q15109 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770958 0.82 PARP1 (0.51) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL15175542 0.75 GRM4 (0.38) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL3716902 0.74 PARP1 (0.44) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL27514150 0.74 GAA (0.53) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3714492 0.73 JAK3 (0.43) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2488255 0.73 PARP1 (0.53) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3714860 0.72 KCNA5 (0.49) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2713150 0.72 JAK3 (0.45) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL447126 0.72 NAPRT (0.68) PARP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL28905992 0.72 P2RX7 (0.65) PARP1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743794-B2 MULTIDRUG RESISTANCE PROTEIN; CANCER; 3-(9-CHLORO-3-METHYL-4-OXO-5H-ISOXAZOLO(4,3-C)QUINOLIN-5-YL)) CYCLOHEXYL)-2-PIPERIDYLACETAMIDE ELI LILLY AND COMPANY 2004-06-01 US disclosed