SCHEMBL6801979

SCHEMBL6801979

CC(=O)N(Cc1ccc(O)cc1)c1ccc(O)cc1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 3/20 0.53
TSPO P30536 5/20 0.51
PDK2 Q15119 2/20 0.50
PDK4 Q16654 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
PDK1 Q15118 1/20 0.50
PDK3 Q15120 1/20 0.50
ESR1 P03372 2/20 0.46
ESR2 Q92731 2/20 0.46
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6799498 0.87 TSPO (0.51) LTB4R2TSPOPDK2PDK4CYP3A4
SCHEMBL10926482 0.80 ALDH1A1 (0.48) CYP3A4ESR1ESR2ALDH1A1
SCHEMBL27872334 0.78 ESR1 (0.40) PDK2PDK4CYP3A4CYP2C9PDK1
SCHEMBL9645342 0.78 ESR1 (0.40) PDK2PDK4CYP3A4CYP2C9PDK1
SCHEMBL5694553 0.78 TSPO (0.72) LTB4R2TSPOALDH1A1
SCHEMBL9416644 0.78 ALDH1A1 (0.50) CYP3A4ESR1ESR2ALDH1A1
SCHEMBL1259310 0.77 PDK1 (0.58) LTB4R2PDK2PDK4PDK1ESR1
SCHEMBL935744 0.77 MLYCD (0.41) ESR1ESR2ALDH1A1
SCHEMBL29588899 0.77 ESR1 (0.42) LTB4R2PDK2PDK4CYP3A4CYP2C9
SCHEMBL20219028 0.77 TSPO (0.69) LTB4R2TSPOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1308297-C Phenyl sulfamate derivs. TEIKOKU HORMONE MFG CO LTD (JP) 2007-04-04 CN disclosed
US-6762205-B1 STEROID SULFATASE INHIBITORS WITHOUT ESTROGENIC SIDE EFFECT ACTION TEIKOKU HORMONE MFG. CO., LTD. (JP) 2004-07-13 US disclosed
CN-1360570-A Phenyl sulfamate derivs. TEIKOKU HORMONE MFG CO LTD (JP) 2002-07-24 CN disclosed
EP-1193250-A1 PHENYL SULFAMATE DERIVATIVES Teikoku Hormone Mfg. Co., Ltd. (JP) 2002-04-03 EP disclosed