SCHEMBL6802695

SCHEMBL6802695

COc1cccc(OC)c1C(=O)Nc1ccc(CC(NC(=O)N2CCC(n3c(=O)[nH]c4ccccc43)CC2)C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 15/20 0.61
CYP3A4 P08684 7/20 0.57
ALDH1A1 P00352 1/20 0.55
OPRM1 P35372 1/20 0.51
RAMP1 O60894 1/20 0.51
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
PLD2 O14939 1/20 0.48
PLD1 Q13393 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802711 0.90 CALCRL (0.63) CALCRLCYP3A4ALDH1A1OPRM1RAMP1
SCHEMBL6808345 0.89 CALCRL (0.63) CALCRLCYP3A4ALDH1A1OPRM1RAMP1
SCHEMBL6808589 0.84 CALCRL (0.52) CALCRLCYP3A4ALDH1A1RAMP1DRD2
SCHEMBL6807923 0.77 CTSB (0.48) CALCRLALDH1A1PLD2PLD1
SCHEMBL4698559 0.76 CALCRL (0.65) CALCRLCYP3A4ALDH1A1OPRM1RAMP1
SCHEMBL4698557 0.76 CALCRL (0.65) CALCRLCYP3A4ALDH1A1OPRM1RAMP1
SCHEMBL3963833 0.76 CALCRL (0.81) CALCRLCYP3A4ALDH1A1RAMP1
SCHEMBL6807110 0.74 ITGA4 (0.47) ALDH1A1
SCHEMBL6812351 0.74 CALCRL (0.52) CALCRLCYP3A4ALDH1A1RAMP1
SCHEMBL22869715 0.74 HSD11B1 (0.73) ALDH1A1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient TORAY INDUSTRIES, INC. (JP) 2004-02-26 US disclosed
EP-1323709-A1 UREA DERIVATIVE AND ADHESIVE-MOLECULE INHIBITOR CONTAINING THE SAME AS ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2003-07-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039040-A1 Urea derivative and adhesive-molecule inhibitor containing the same as active ingredient ICAM1, VCAM1, EPCAM CALCRL 1811/4885CYP3A4 3783/4885ALDH1A1 283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.