SCHEMBL6802996

SCHEMBL6802996

CNC(=O)c1cc(-c2ccc(O)cc2)on1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.68
NPC1 O15118 7/20 0.66
RAB9A P51151 7/20 0.66
ALDH1A1 P00352 4/20 0.66
HDAC3 O15379 1/20 0.62
HDAC4 P56524 1/20 0.62
HDAC1 Q13547 1/20 0.62
HDAC7 Q8WUI4 1/20 0.62
HDAC2 Q92769 1/20 0.62
HDAC10 Q969S8 1/20 0.62
HDAC11 Q96DB2 1/20 0.62
HDAC8 Q9BY41 1/20 0.62
HDAC6 Q9UBN7 1/20 0.62
HDAC9 Q9UKV0 1/20 0.62
HDAC5 Q9UQL6 1/20 0.62
MLLT1 Q03111 1/20 0.62
TSHR P16473 1/20 0.61
KMT2A Q03164 2/20 0.60
POLB P06746 2/20 0.60
HPGD P15428 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3219488 0.86 RAB9A (0.72) TP53NPC1RAB9AALDH1A1KMT2A
SCHEMBL10153708 0.85 ALDH1A1 (0.67) NPC1RAB9AALDH1A1KMT2AHPGD
SCHEMBL21446983 0.84 ROCK2 (0.59) TP53NPC1RAB9AALDH1A1MLLT1
SCHEMBL22322454 0.84 HPGD (0.55) TP53NPC1RAB9AALDH1A1KMT2A
SCHEMBL15196594 0.81 ALDH1A1 (0.72) TP53NPC1RAB9AALDH1A1HDAC3
SCHEMBL19245571 0.80 ROCK2 (0.57) TP53NPC1RAB9AALDH1A1HDAC6
SCHEMBL72786 0.80 ALDH1A1 (1.00) TP53NPC1RAB9AALDH1A1HDAC3
SCHEMBL21536740 0.78 ALDH1A1 (0.62) TP53NPC1RAB9AALDH1A1HDAC4
SCHEMBL17732022 0.78 ALDH1A1 (0.72) TP53NPC1RAB9AALDH1A1TSHR
SCHEMBL3236082 0.78 ROCK2 (0.49) TP53NPC1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6762205-B1 STEROID SULFATASE INHIBITORS WITHOUT ESTROGENIC SIDE EFFECT ACTION TEIKOKU HORMONE MFG. CO., LTD. (JP) 2004-07-13 US disclosed
EP-1193250-A1 PHENYL SULFAMATE DERIVATIVES Teikoku Hormone Mfg. Co., Ltd. (JP) 2002-04-03 EP disclosed