SCHEMBL6804734

SCHEMBL6804734

NC(=O)c1cccc2nc(-c3cnn(-c4ccc(Br)cc4)c3)[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.42
NR2E3 Q9Y5X4 1/20 0.42
MAP4K4 O95819 3/20 0.39
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA9 Q16790 3/20 0.38
CA2 P00918 2/20 0.38
TYK2 P29597 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
PLK4 O00444 2/20 0.36
PRKX P51817 2/20 0.36
ROCK1 Q13464 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
DAPK3 O43293 1/20 0.36
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806401 0.90 GRM2 (0.52) GRM2NR2E3MAP4K4ADORA2AADORA2B
SCHEMBL6810614 0.89 MAP4K4 (0.52) GRM2NR2E3MAP4K4ADORA2AADORA2B
SCHEMBL6804729 0.83 PARP1 (0.57) MAP4K4PLK4PRKXROCK1CLK4
SCHEMBL6801835 0.82 AURKB (0.44) MAP4K4PLK4PRKXROCK1CLK4
SCHEMBL6803965 0.80 EPHX2 (0.55) GRM2MAP4K4PLK4PRKXROCK1
SCHEMBL6807217 0.77 JAK3 (0.42) MAP4K4TYK2PLK4PRKXROCK1
SCHEMBL3579908 0.74 PARP1 (0.61) MAP4K4PLK4PRKXROCK1CLK4
SCHEMBL6806394 0.73 PARP1 (0.67) MAP4K4PLK4PRKXROCK1CLK4
SCHEMBL6810606 0.72 PARP1 (0.69) MAP4K4PLK4PRKXROCK1CLK4
SCHEMBL6586796 0.72 PKN1 (0.39) NR2E3MAP4K4PLK4PRKXROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed