SCHEMBL6801835

SCHEMBL6801835

NC(=O)c1cccc2nc(-c3ccn(-c4ccc(Br)cc4)c3)[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.44
KDR P35968 2/20 0.44
PARP1 P09874 12/20 0.36
CHEK2 O96017 2/20 0.35
TNKS O95271 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
PLK4 O00444 2/20 0.35
MAP4K4 O95819 2/20 0.35
PRKX P51817 2/20 0.35
ROCK1 Q13464 2/20 0.35
CLK4 Q9HAZ1 2/20 0.35
PKN1 Q16512 2/20 0.35
PKN2 Q16513 2/20 0.35
MAPK13 O15264 1/20 0.35
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
RPS6KA5 O75582 1/20 0.35
PRKD3 O94806 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807111 0.89 PARP1 (0.46) AURKBKDRPARP1CHEK2TNKS
SCHEMBL6804968 0.86 PARP1 (0.49) AURKBKDRPARP1CHEK2TNKS
SCHEMBL6801829 0.83 AURKB (0.60) AURKBKDRPARP1CHEK2PLK4
SCHEMBL6804734 0.82 GRM2 (0.42) AURKBKDRPARP1CHEK2TNKS
SCHEMBL6807301 0.81 PARP1 (0.39) AURKBKDRPARP1CHEK2PLK4
SCHEMBL3581925 0.81 AURKB (0.47) AURKBKDRPARP1CHEK2PLK4
SCHEMBL3582143 0.81 AURKB (0.56) AURKBKDRPARP1DHODHAURKA
SCHEMBL3575391 0.79 DHODH (0.47) AURKBKDRPARP1CHEK2PLK4
SCHEMBL6804756 0.78 PARP1 (0.37) AURKBKDRPARP1CHEK2PLK4
SCHEMBL6806674 0.76 PARP1 (0.39) AURKBKDRPARP1CHEK2PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed