SCHEMBL6806401

SCHEMBL6806401

NC(=O)c1cccc2nc(-c3cnn(-c4ccccc4)c3)[nH]c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.52
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
PARP1 P09874 6/20 0.45
TYK2 P29597 1/20 0.45
PARP2 Q9UGN5 1/20 0.45
PARP3 Q9Y6F1 1/20 0.45
NR2E3 Q9Y5X4 1/20 0.44
DHODH Q02127 1/20 0.41
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
NFKB1 P19838 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
HPGDS O60760 1/20 0.40
ALKBH2 Q6NS38 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804734 0.90 GRM2 (0.42) GRM2ADORA2AADORA2BADORA1PARP1
SCHEMBL6810614 0.90 MAP4K4 (0.52) GRM2ADORA2AADORA2BADORA1PARP1
SCHEMBL6803965 0.82 EPHX2 (0.55) GRM2PARP1PARP2KCNH2MAP4K4
SCHEMBL6806394 0.82 PARP1 (0.67) PARP1PARP2DHODHMAP4K4PLK4
SCHEMBL3579908 0.81 PARP1 (0.61) PARP1PARP2DHODHNPC1HPGD
SCHEMBL6807217 0.80 JAK3 (0.42) PARP1TYK2MAP4K4PLK4CHEK1
SCHEMBL6810590 0.76 GRM2 (0.54) GRM2PARP1NPC1MAPTRAB9A
SCHEMBL6805042 0.75 AURKA (0.57) PARP1NPC1MAPTHPGDNFKB1
SCHEMBL6809996 0.74 PKN1 (0.63) PARP1PARP2DHODHMAPTHPGD
SCHEMBL2149454 0.74 PARP1 (0.63) PARP1PARP2DHODHMAP4K4PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed