SCHEMBL6804968

SCHEMBL6804968

COc1ccc(-n2ccc(-c3nc4cccc(C(N)=O)c4[nH]3)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.49
PLA2G2A P14555 1/20 0.49
ALOX15 P16050 1/20 0.49
PTGS2 P35354 1/20 0.49
CHEK2 O96017 5/20 0.43
KDR P35968 1/20 0.42
AURKB Q96GD4 1/20 0.42
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TNKS O95271 1/20 0.38
GUSB P08236 1/20 0.38
CASP3 P42574 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
BRD4 O60885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801835 0.86 AURKB (0.44) PARP1CHEK2KDRAURKBTNKS
SCHEMBL6807111 0.86 PARP1 (0.46) PARP1CHEK2KDRAURKBTNKS
SCHEMBL6804961 0.84 PARP1 (0.72) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL6807301 0.81 PARP1 (0.39) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL3582143 0.78 AURKB (0.56) PARP1KDRAURKB
SCHEMBL3581925 0.78 AURKB (0.47) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL31053400 0.78 PARP1 (0.67) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL3575391 0.77 DHODH (0.47) PARP1ALOX15CHEK2KDRAURKB
SCHEMBL6806674 0.76 PARP1 (0.39) PARP1PLA2G2AALOX15PTGS2CHEK2
SCHEMBL6804756 0.76 PARP1 (0.37) PARP1CHEK2KDRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed