SCHEMBL6807301

SCHEMBL6807301

Cc1cccc(C)c1-n1ccc(-c2nc3cccc(C(N)=O)c3[nH]2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.39
CHEK2 O96017 2/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
AURKB Q96GD4 2/20 0.37
KDR P35968 1/20 0.37
EPHB4 P54760 1/20 0.36
PLK4 O00444 1/20 0.36
MAPK13 O15264 1/20 0.36
DYRK3 O43781 1/20 0.36
ROCK2 O75116 1/20 0.36
RPS6KA5 O75582 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PIM1 P11309 1/20 0.36
PHKG2 P15735 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CSNK1D P48730 1/20 0.36
CLK2 P49760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807298 0.82 PARP1 (0.60) PARP1CHEK2AURKBPLK4MAPK13
SCHEMBL6807111 0.81 PARP1 (0.46) PARP1CHEK2AURKBKDRPLK4
SCHEMBL6801835 0.81 AURKB (0.44) PARP1CHEK2AURKBKDRPLK4
SCHEMBL6804968 0.81 PARP1 (0.49) PARP1CHEK2AURKBKDRPLA2G2A
SCHEMBL6806674 0.80 PARP1 (0.39) PARP1CHEK2AURKBKDRPLK4
SCHEMBL6804756 0.79 PARP1 (0.37) PARP1CHEK2AURKBKDRPLK4
SCHEMBL3579908 0.75 PARP1 (0.61) PARP1CHEK2AURKBPLK4MAPK13
SCHEMBL29696369 0.75 NPC1 (0.53) PARP1CYP3A4CYP2C9CSNK1DDHODH
SCHEMBL6804607 0.74 PARP1 (0.45) PARP1AURKBKDRDYRK3PRKD3
SCHEMBL6803965 0.74 EPHX2 (0.55) PARP1KDRPLK4ROCK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed