SCHEMBL6806674

SCHEMBL6806674

CC(C)(C)n1ccc(-c2nc3cccc(C(N)=O)c3[nH]2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.39
PLK4 O00444 2/20 0.37
MAP4K4 O95819 2/20 0.37
PRKX P51817 2/20 0.37
ROCK1 Q13464 2/20 0.37
CLK4 Q9HAZ1 2/20 0.37
PKN1 Q16512 2/20 0.37
PKN2 Q16513 2/20 0.37
MAPK13 O15264 1/20 0.37
DYRK3 O43781 1/20 0.37
ROCK2 O75116 1/20 0.37
RPS6KA5 O75582 1/20 0.37
PRKD3 O94806 1/20 0.37
CHEK2 O96017 1/20 0.37
PIM1 P11309 1/20 0.37
PHKG2 P15735 1/20 0.37
PRKACA P17612 1/20 0.37
RPS6KB1 P23443 1/20 0.37
CSNK1D P48730 1/20 0.37
CLK2 P49760 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806672 0.81 PARP1 (0.62) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL6807217 0.81 JAK3 (0.42) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL6807301 0.80 PARP1 (0.39) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL3579908 0.77 PARP1 (0.61) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL6801835 0.76 AURKB (0.44) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL6807111 0.76 PARP1 (0.46) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL6804968 0.76 PARP1 (0.49) PARP1CHEK2AURKBPLA2G2AALOX15
SCHEMBL6804607 0.76 PARP1 (0.45) PARP1MAP4K4CLK4PKN2DYRK3
SCHEMBL6803965 0.76 EPHX2 (0.55) PARP1PLK4MAP4K4PRKXROCK1
SCHEMBL7583436 0.76 PARP1 (0.66) PARP1PLK4MAP4K4PRKXROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed