SCHEMBL6806583

SCHEMBL6806583

CC(=O)n1cc(-c2nc3c(C(N)=O)cccc3[nH]2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.57
DHODH Q02127 3/20 0.53
PLK4 O00444 1/20 0.50
MAPK13 O15264 1/20 0.50
DYRK3 O43781 1/20 0.50
ROCK2 O75116 1/20 0.50
RPS6KA5 O75582 1/20 0.50
PRKD3 O94806 1/20 0.50
MAP4K4 O95819 1/20 0.50
CHEK2 O96017 1/20 0.50
PIM1 P11309 1/20 0.50
PHKG2 P15735 1/20 0.50
PRKACA P17612 1/20 0.50
RPS6KB1 P23443 1/20 0.50
CSNK1D P48730 1/20 0.50
CLK2 P49760 1/20 0.50
GSK3A P49840 1/20 0.50
PRKX P51817 1/20 0.50
PRKCZ Q05513 1/20 0.50
STK3 Q13188 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806945 0.87 PARP1 (0.60) PARP1DHODHPLK4MAPK13DYRK3
SCHEMBL6587773 0.84 PARP1 (0.46) PARP1
SCHEMBL6806586 0.83 HTT (0.46) PARP1
SCHEMBL6810278 0.78 PIM1 (0.54) PARP1DHODHPRKD3MAP4K4PIM1
SCHEMBL6801381 0.78 L3MBTL1 (0.51) PARP1DHODH
SCHEMBL6802028 0.76 PARP1 (0.66) PARP1DHODHPLK4MAPK13DYRK3
SCHEMBL29411925 0.75 PARP1 (0.72) PARP1DHODHPLK4MAPK13DYRK3
SCHEMBL6805760 0.75 PARP1 (0.51) PARP1DHODH
Hydrochloric Acid SCHEMBL6809753 0.73 PARP1 (0.60) PARP1DHODHPLK4MAPK13DYRK3
SCHEMBL29411891 0.73 PARP1 (1.00) PARP1DHODHPLK4MAPK13DYRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed