SCHEMBL6587773

SCHEMBL6587773

CC(=O)n1cc(-c2nc3c(OC(N)=O)cccc3[nH]2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.46
HTT P42858 2/20 0.43
CREBBP Q92793 4/20 0.42
BRD9 Q9H8M2 2/20 0.42
BRPF1 P55201 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PDE5A O76074 1/20 0.40
GAA P10253 1/20 0.37
HPSE Q9Y251 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6586959 0.88 KDM4E (0.56) PARP1HTTSMN1; SMN2KDM4ENPC1
SCHEMBL6806583 0.84 PARP1 (0.57) PARP1
SCHEMBL6589817 0.80 PIM1 (0.41) PARP1HTTSMN1; SMN2KDM4ENPC1
SCHEMBL6590569 0.80 L3MBTL1 (0.48) PARP1KDM4E
SCHEMBL6588173 0.77 PARP1 (0.49) PARP1ALDH1A1PDE5AHPSEMEN1
SCHEMBL17023492 0.76 CREBBP (0.48) HTTCREBBPBRD9BRPF1SMN1; SMN2
SCHEMBL6587182 0.74 MEN1 (0.52) PARP1SMN1; SMN2KDM4EALDH1A1LMNA
SCHEMBL7479706 0.73 PARP1 (0.49) PARP1PDE5AGAAHPSE
SCHEMBL6588299 0.72 PARP1 (0.47) PARP1SMN1; SMN2NPC1ALDH1A1MAPT
SCHEMBL6806586 0.72 HTT (0.46) PARP1HTTCREBBPBRD9BRPF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed