SCHEMBL680683

SCHEMBL680683

COC(=O)c1ccc[nH]c1=O

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.60
KDM4E B2RXH2 5/20 0.53
GAA P10253 2/20 0.53
GLA P06280 1/20 0.53
TSHR P16473 2/20 0.50
MAPT P10636 1/20 0.50
MAPK1 P28482 1/20 0.50
LMNA P02545 1/20 0.50
NR4A2 P43354 1/20 0.50
CREBBP Q92793 1/20 0.50
ALDH1A1 P00352 2/20 0.48
CFTR P13569 1/20 0.48
HSD17B10 Q99714 1/20 0.48
RECQL P46063 1/20 0.48
POLB P06746 1/20 0.47
ATM Q13315 1/20 0.47
TYK2 P29597 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4428793 0.98 NAPRT (0.58) NAPRTKDM4EGAAGLATSHR
SCHEMBL14632936 0.80 NAPRT (0.55) NAPRTKDM4EGAATSHRMAPT
SCHEMBL930113 0.80 TSHR (0.61) NAPRTKDM4EGAATSHRMAPT
SCHEMBL8679491 0.80 NAPRT (0.55) NAPRTKDM4EGAATSHRMAPT
Hydrochloric Acid SCHEMBL4428342 0.79 TSHR (0.59) NAPRTKDM4EGAATSHRMAPT
Dimethyl Phthalate SCHEMBL29850852 0.78 FKBP5 (0.57) KDM4EGAAGLATSHRMAPT
SCHEMBL3182033 0.78 NAPRT (0.67) NAPRTKDM4EGAATSHRMAPT
SCHEMBL29532188 0.78 PARP1 (0.53) KDM4EGAALMNANR4A2CREBBP
SCHEMBL22230076 0.78 PARP1 (0.53) KDM4EGAALMNANR4A2CREBBP
SCHEMBL425117 0.77 NAPRT (0.72) NAPRTKDM4EGAATSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 228 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4698517-A1 <SUP2/>? <SUB2/>?4?NOVEL COMPOUNDS AS ?? <NS1:SUB>7</NS1:SUB>?INHIBITORS Evotec International GmbH (DE) 2026-02-25 EP disclosed
US-20260042765-A1 PYRROLOTRIAZINE COMPOUNDS AS TAM INHIBITORS INCYTE CORP (US) 2026-02-12 US disclosed
US-20250361223-A1 AMIDE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LTD (CN) 2025-11-27 US disclosed
US-12435062-B2 Amide compounds and uses thereof HUTCHISON MEDIPHARMA LIMITED (CN) 2025-10-07 US disclosed
US-12415809-B2 Pyrrolotriazine compounds as tam inhibitors INCYTE CORPORATION (US) 2025-09-16 US disclosed
EP-4573085-A1 SUBSTITUTED PYRIDINONE COMPOUNDS AS CBL-B INHIBITORS Glenmark Pharmaceuticals Limited (IN) 2025-06-25 EP disclosed
WO-2025072462-A1 SULFONAMIDE DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS NIKANG THERAPEUTICS, INC. (US) 2025-04-03 WO disclosed
WO-2025061180-A1 NITROGEN-CONTAINING CYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 杭州多域生物技术有限公司 2025-03-27 WO disclosed
CN-119546587-A Substituted pyridone compounds as CBL-B inhibitors 格兰玛克制药有限公司 2025-02-28 CN disclosed
US-20250066360-A1 PYRIDINE-CONTAINING POLYCYCLIC DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF JIANGSU HANSOH PHARMACEUTICAL GROUP CO., LTD. (CN) 2025-02-27 US disclosed
WO-2007103308-A2 HETEROBICYCLIC PYRAZOLE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-09-13 WO disclosed
WO-2007103308-A2 HETEROBICYCLIC PYRAZOLE COMPOUNDS AND METHODS OF USE ARRAY BIOPHARMA INC. (US) 2007-09-13 WO disclosed
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. 2007-08-23 US disclosed
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. 2007-08-23 US disclosed
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. 2007-08-23 US disclosed
EP-0265126-B1 Process for the preparation of fused pyridine compounds UNIV PRINCETON (US) 1994-04-13 EP disclosed
US-4988813-A Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-01-29 US disclosed
US-4902796-A 6-alkenyl and ethynyl derivatives of 2-amino-4-hydroxypyrido[2,3-d]pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1990-02-20 US disclosed
US-4818819-A Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-04-04 US disclosed
EP-0265126-A2 Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1988-04-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ERBB2, LCK, SRC NAPRT 1872/4885KDM4E 3968/4885GAA 1103/4885
US-20260042765-A1 PYRROLOTRIAZINE COMPOUNDS AS TAM INHIBITORS MAP2K2, TTK, MAP2K5 NAPRT 1219/4885KDM4E 212/4885GAA 3285/4885
US-12435062-B2 Amide compounds and uses thereof ASNS, ASS1, NAT1 NAPRT 283/4885KDM4E 1449/4885GAA 374/4885
US-20250361223-A1 AMIDE COMPOUNDS AND USES THEREOF ASNS, NAT1, AADAC NAPRT 215/4885KDM4E 1690/4885GAA 381/4885
US-12415809-B2 Pyrrolotriazine compounds as tam inhibitors MERTK, MAP3K15, MAP3K5 NAPRT 704/4885KDM4E 769/4885GAA 1385/4885
US-20250066360-A1 PYRIDINE-CONTAINING POLYCYCLIC DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF MYD88, NOD1, LITAF NAPRT 1775/4885KDM4E 1386/4885GAA 2987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.