SCHEMBL6806909

SCHEMBL6806909

COc1nc(N(C)C)c2ccccc2c1-c1nc2cccc(C(N)=O)c2[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 2/20 0.38
HSD17B10 Q99714 2/20 0.38
LMNA P02545 1/20 0.38
PARP1 P09874 13/20 0.38
PDE4B Q07343 1/20 0.37
GRM2 Q14416 1/20 0.36
ALOX15 P16050 2/20 0.36
PLA2G2A P14555 1/20 0.36
PTGS2 P35354 1/20 0.36
CDK9 P50750 1/20 0.36
DYRK1A Q13627 1/20 0.36
PDGFRB P09619 1/20 0.35
FGFR1 P11362 1/20 0.35
KDR P35968 1/20 0.35
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6806906 0.84 PARP1 (0.56) PARP1ALOX15PLA2G2APTGS2DYRK1A
SCHEMBL6585078 0.75 PARP1 (0.44) ALDH1A1HSD17B10PARP1ALOX15PLA2G2A
SCHEMBL6806330 0.73 MEN1 (0.60) KDM4EALDH1A1HSD17B10LMNAPARP1
SCHEMBL8648025 0.73 PARP1 (0.67) PARP1CDK9DYRK1AFGFR1
SCHEMBL3579908 0.70 PARP1 (0.61) KDM4EALDH1A1PARP1DYRK1ACLK4
SCHEMBL31053400 0.70 PARP1 (0.67) PARP1ALOX15PLA2G2APTGS2CLK4
SCHEMBL17048129 0.69 KDM4E (0.56) KDM4EALDH1A1HSD17B10PARP1DYRK1A
SCHEMBL6806564 0.68 ADORA3 (0.54) PARP1FGFR1KDRCLK4
SCHEMBL6802033 0.68 FGFR1 (0.51) KDM4EALDH1A1LMNAPARP1FGFR1
SCHEMBL6805414 0.68 PLK4 (0.39) PARP1FGFR1KDRCLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6696437-B1 Heterocyclically substituted benzimidazoles, the production and application thereof ABBOTT GMBH & CO. KG (DE) 2004-02-24 US disclosed