SCHEMBL681240

SCHEMBL681240

C=C(C(C)C)[C@H](CCNCC(N)=O)c1ccc(Br)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.41
CYP1A2 P05177 1/20 0.36
EPHX1 P07099 2/20 0.35
CNR1 P21554 1/20 0.34
F2 P00734 1/20 0.34
F7 P08709 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
HSP90AA1 P07900 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL681056 0.88 ALOX5 (0.42) ALOX5CYP1A2EPHX1CNR1F2
SCHEMBL12188504 0.85 CYP1A2 (0.41) ALOX5CYP1A2EPHX1CNR1F2
SCHEMBL2738521 0.85 ALOX5 (0.40) ALOX5CYP1A2EPHX1CNR1SMN1; SMN2
SCHEMBL681418 0.82 ALDH1A1 (0.36) ALOX5CYP1A2CNR1SMN1; SMN2KMT2A
SCHEMBL681806 0.79 CYP1A2 (0.37) ALOX5CYP1A2CNR1SMN1; SMN2ALDH1A1
SCHEMBL680223 0.77 ALOX5 (0.42) ALOX5CYP1A2EPHX1SMN1; SMN2KMT2A
SCHEMBL681301 0.77 ALOX5 (0.31) ALOX5CYP1A2
SCHEMBL17803820 0.76 PKM (0.39) ALOX5CYP1A2GAAHTT
SCHEMBL680150 0.74 HTR2A (0.43) ALOX5CYP1A2EPHX1SMN1; SMN2KMT2A
SCHEMBL681405 0.73 ALOX5 (0.38) ALOX5CYP1A2CNR1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9359340-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2016-06-07 US disclosed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed