SCHEMBL6814812

SCHEMBL6814812

CC(C)(C)c1ccc(-c2cncc(C(=O)Nc3ccc(C#N)cc3C(=O)OC(=O)c3cc(C#N)ccc3NC(=O)c3cncc(-c4ccccc4C(F)(F)F)c3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
SAE1 Q9UBE0 1/20 0.46
UBA2 Q9UBT2 1/20 0.46
NR1H4 Q96RI1 1/20 0.45
SCN10A Q9Y5Y9 2/20 0.43
KCNH2 Q12809 1/20 0.43
XDH P47989 1/20 0.43
UBE2N P61088 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CTSA P10619 1/20 0.41
PAX8 Q06710 1/20 0.40
ABL1 P00519 2/20 0.40
TP53 P04637 1/20 0.40
TRPV1 Q8NER1 3/20 0.39
RXFP1 Q9HBX9 1/20 0.39
PIK3CA P42336 1/20 0.38
KDM1A O60341 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6834009 0.83 CTSA (0.47) KDM4EMAPTSAE1UBA2SCN10A
SCHEMBL6830649 0.81 KCNH2 (0.54) KDM4EMAPTSAE1UBA2NR1H4
SCHEMBL6833875 0.77 KDM4E (0.52) KDM4EMAPTSAE1UBA2SCN10A
SCHEMBL6833755 0.73 KCNH2 (0.55) KDM4EMAPTSAE1UBA2SCN10A
SCHEMBL6835793 0.72 KCNH2 (0.49) NR1H4SCN10AKCNH2XDHKMT2A
SCHEMBL6833154 0.72 KDM4E (0.54) KDM4EMAPTSAE1UBA2SCN10A
SCHEMBL6357270 0.71 SERPINE1 (0.62) MAPTNR1H4KMT2ATDP1
SCHEMBL1317262 0.70 ACLY (0.52) CTSAHDAC1AXL
SCHEMBL6834158 0.70 XDH (0.54) KDM4EMAPTSAE1UBA2SCN10A
SCHEMBL1317261 0.69 CTSA (0.46) SCN10AKCNH2CTSAABL1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004018428-A1 ANTIBACTERIAL BENZOIC ACID DERIVATIVES PHARMACIA & UPJOHN COMPANY LLC (US) 2004-03-04 WO disclosed